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Found 6 of affinity data for UniProtKB/TrEMBL: Q63645
TargetProteinase-activated receptor 2(RAT)
The University of Calgary

Curated by PDSP Ki Database
LigandPNGBDBM85517(CAS_171436-38-7 | SL-NH2 | SLIGRL-NH2)
Affinity DataKi:  260nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProteinase-activated receptor 2(RAT)
The University of Calgary

Curated by PDSP Ki Database
LigandPNGBDBM85518(tc-NH2 | trans-cinnamoyl-LIGRLO-NH2)
Affinity DataKi:  260nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProteinase-activated receptor 2(RAT)
The University of Calgary

Curated by PDSP Ki Database
LigandPNGBDBM85516(CAS_141923-41-3 | P5-NH2 | SFLLR-NH2)
Affinity DataKi:  2.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProteinase-activated receptor 2(RAT)
The University of Calgary

Curated by PDSP Ki Database
LigandPNGBDBM85088(SFLLR-OH)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProteinase-activated receptor 2(RAT)
The University of Calgary

Curated by PDSP Ki Database
LigandPNGBDBM50440871(CHEMBL2431725)
Affinity DataIC50:  5.00E+4nMAssay Description:Antagonist activity at rat PAR2 expressed in rat KNRK cells assessed as inhibition of trypsin-induced receptor activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(RAT)
The University of Calgary

Curated by PDSP Ki Database
LigandPNGBDBM50440870(CHEMBL2431726)
Affinity DataIC50:  5.00E+4nMAssay Description:Antagonist activity at rat PAR2 expressed in rat KNRK cells assessed as inhibition of trypsin-induced receptor activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed